1信号转导与转录激活因子3(STAT3)抑制剂及其抗肿瘤研究进展1
Progress in the Research of STAT3 Inhibitors as Anticancer Agents
余文颖李洋孔令义
2选择性EGFR T790M抑制剂的研究进展17
Recent Advance on the Discovery of T790M Mutantselective EGFR Inhibitors
徐石林徐田锋丁克3FLT
3ITD及其抑制剂的研究进展38
Advances in FLT3 Internal Tandem Duplications Mutation and Inhibitors of FLT3ITD
钟杭蔡婷赵临襄
4组蛋白去甲基化酶及其抑制剂的研究进展57
Progress in the Research of Histone Demethylases and Their Inhibitors
郑一超刘宏民
5 组蛋白去乙酰化酶抑制剂研究进展77
Progress in Histone Deacetylase Inhibitors
安娜高明邓卫平
6NAD+依赖的组蛋白去乙酰化酶Sirtuin激活剂与抑制剂的研究进展107
Progress in NAD+dependent Sirtuins Activators and Inhibitors
王磊方浩
7靶向IKKβ激酶抑制剂的研究进展120
Progress in Targeting IKKβ Kinase Inhibitors
褚红喜黄婧婕孙昊鹏尤启冬
8缺氧诱导因子HIF介导肿瘤耐药及其相关药物的研究进展131
The Research Development of Hypoxiamediated Drug Resistance and Drug Candidates
陈亚琼彭晖
9天然萜类化合物逆转肿瘤和细菌多药耐药的研究进展159
Progress in the Research of Natural Terpenes as Reversal Agents of Multidrug Resistance in Cancer and Bacteria
张恒源徐进宜
10抗菌肽设计的研究进展179
Recent Studies on Designing Antimicrobial Peptides
张伟谢俊秋张邦治王锐
11治疗糖尿病的新策略——SGLT2抑制剂202
A Novel Strategy for Diabetes TreatmentSGLT2 Inhibitors
王学堃钱海黄文龙
12GPR40 和GPR120调控剂的研究进展225
Progress in GPR40 and GPR120 Modulators
雷显涛温小安孙宏斌
13抗阿尔茨海默病药物研究进展255
Progresses of the Development of antiAlzheimer Drugs
房雷苟少华
14载体转运系统介导的脑靶向药物研究进展281
Progress in Carriermediated Brain Targeting Drugs
吴勇李晓岑海俐
15与重大疾病相关的糖类药物的研究进展303
Progress in the Research of Carbohydratebased Drugs Associated with Major Diseases
王晓丽田光宗汪学彬尹健
16一氧化氮供体偶氮二醇盐的O2保护策略及其应用研究进展321
Research Progress in O2protection and Application of Nitric Oxide Donor Diazeniumdiolates
黄张建赖宜生彭司勋张奕华